A small-molecule modulator interacts directly with deltaPhe508-CFTR to modify its ATPase activity and conformational stability. [electronic resource]
- Molecular pharmacology Jun 2009
- 1430-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1521-0111
10.1124/mol.109.055608 doi
Adenosine Triphosphatases--metabolism Animals Cell Line Cresols--pharmacology Cricetinae Cystic Fibrosis Transmembrane Conductance Regulator--genetics Humans Mutation Protein Binding Protein Conformation Pyrazoles--pharmacology Structure-Activity Relationship