Hall, Adrian Discovery of sodium 6-[(5-chloro-2-phenyl)methyl]-2-pyridinecarboxylate (GSK269984A) an EP(1) receptor antagonist for the treatment of inflammatory pain. [electronic resource] - Bioorganic & medicinal chemistry letters May 2009 - 2599-603 p. digital Publication Type: Journal Article ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2009.02.112 doi Subjects--Topical Terms: Analgesics--chemical synthesisAnimalsCentral Nervous System--drug effectsChemistry, Pharmaceutical--methodsDrug DesignHumansHydrogen-Ion ConcentrationInflammation--drug therapyInhibitory Concentration 50Models, ChemicalNicotinic Acids--chemical synthesisPyridines--chemical synthesisRatsReceptors, Prostaglandin E--antagonists & inhibitorsStructure-Activity Relationship