Duplantier, Allen J

3-Benzyl-1,3-oxazolidin-2-ones as mGluR2 positive allosteric modulators: Hit-to lead and lead optimization. [electronic resource] - Bioorganic & medicinal chemistry letters May 2009 - 2524-9 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2009.03.032 doi


Administration, Oral
Allosteric Regulation
Allosteric Site
Carbamates--chemistry
Chemistry, Pharmaceutical--methods
Drug Design
Humans
Inhibitory Concentration 50
Ligands
Microsomes--metabolism
Models, Chemical
Molecular Structure
Oxazolidinones--chemical synthesis
Receptors, Metabotropic Glutamate--antagonists & inhibitors
Schizophrenia--drug therapy