3-Benzyl-1,3-oxazolidin-2-ones as mGluR2 positive allosteric modulators: Hit-to lead and lead optimization. [electronic resource]
- Bioorganic & medicinal chemistry letters May 2009
- 2524-9 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.03.032 doi
Administration, Oral Allosteric Regulation Allosteric Site Carbamates--chemistry Chemistry, Pharmaceutical--methods Drug Design Humans Inhibitory Concentration 50 Ligands Microsomes--metabolism Models, Chemical Molecular Structure Oxazolidinones--chemical synthesis Receptors, Metabotropic Glutamate--antagonists & inhibitors Schizophrenia--drug therapy