Debenham, John S Pyridopyrimidine based cannabinoid-1 receptor inverse agonists: Synthesis and biological evaluation. [electronic resource] - Bioorganic & medicinal chemistry letters May 2009 - 2591-4 p. digital Publication Type: Journal Article ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2009.03.005 doi Subjects--Topical Terms: Administration, OralAnimalsCannabinoid Receptor AgonistsCannabinoids--chemistryChemistry, Pharmaceutical--methodsDrug DesignHumansInhibitory Concentration 50Obesity--drug therapyProtein Structure, TertiaryPyrimidines--chemistryRatsReceptor, Cannabinoid, CB1--agonistsReceptor, Cannabinoid, CB2--agonistsStructure-Activity Relationship