Rational mutagenesis to support structure-based drug design: MAPKAP kinase 2 as a case study. [electronic resource]
- BMC structural biology Mar 2009
- 16 p. digital
Publication Type: Journal Article
1472-6807
10.1186/1472-6807-9-16 doi
Amino Acid Substitution Computer Simulation Crystallization Crystallography, X-Ray Drug Design Humans Intracellular Signaling Peptides and Proteins--chemistry Isoenzymes--biosynthesis Mutagenesis, Site-Directed Protein Conformation Protein Kinase Inhibitors--chemistry Protein Serine-Threonine Kinases--biosynthesis