Investigation of the micellar effect of pluronic P85 on P-glycoprotein inhibition: cell accumulation and equilibrium dialysis studies. [electronic resource]
- Journal of pharmaceutical sciences Nov 2009
- 4170-90 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1520-6017
10.1002/jps.21723 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Acridines--pharmacology Animals Biological Transport, Active--drug effects Cell Line Cell-Free System Cells--metabolism Dialysis Dideoxynucleosides--metabolism Diphenylhexatriene--metabolism Dogs Dose-Response Relationship, Drug Drug Resistance, Multiple--drug effects Fluorescent Dyes--metabolism HIV-1--enzymology Inhibitory Concentration 50 Mannitol--immunology Micelles Nelfinavir--metabolism Permeability Poloxamer--pharmacology Protease Inhibitors--pharmacology Saquinavir--metabolism Surface-Active Agents--pharmacology Temperature Tetrahydroisoquinolines--pharmacology Time Factors