Shaik, Naveed

Investigation of the micellar effect of pluronic P85 on P-glycoprotein inhibition: cell accumulation and equilibrium dialysis studies. [electronic resource] - Journal of pharmaceutical sciences Nov 2009 - 4170-90 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1520-6017

10.1002/jps.21723 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Acridines--pharmacology
Animals
Biological Transport, Active--drug effects
Cell Line
Cell-Free System
Cells--metabolism
Dialysis
Dideoxynucleosides--metabolism
Diphenylhexatriene--metabolism
Dogs
Dose-Response Relationship, Drug
Drug Resistance, Multiple--drug effects
Fluorescent Dyes--metabolism
HIV-1--enzymology
Inhibitory Concentration 50
Mannitol--immunology
Micelles
Nelfinavir--metabolism
Permeability
Poloxamer--pharmacology
Protease Inhibitors--pharmacology
Saquinavir--metabolism
Surface-Active Agents--pharmacology
Temperature
Tetrahydroisoquinolines--pharmacology
Time Factors