3-Hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylates--a new class of HIV-1 integrase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Apr 2009
- 1930-4 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.02.055 doi
Animals HIV Integrase--metabolism HIV Integrase Inhibitors--chemical synthesis HIV-1--drug effects Pyrimidines--chemical synthesis Rats Structure-Activity Relationship