DeVore, N M

Key residues controlling binding of diverse ligands to human cytochrome P450 2A enzymes. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Jun 2009 - 1319-27 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1521-009X

10.1124/dmd.109.026765 doi


Amino Acid Sequence
Amino Acid Substitution
Aryl Hydrocarbon Hydroxylases--chemistry
Catalytic Domain--drug effects
Cytochrome P-450 CYP2A6
Cytochrome P-450 Enzyme System--chemistry
Humans
Ligands
Microsomes, Liver
Models, Molecular
Mutagenesis, Site-Directed
Protein Binding--genetics
Protein Conformation
Steroid Hydroxylases--chemistry
Structure-Activity Relationship
Substrate Specificity