1,3,4-Oxadiazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 2: SAR of the C5 position. [electronic resource]
- Bioorganic & medicinal chemistry letters Mar 2009
- 1807-10 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.01.089 doi
Amino Acid Motifs Anti-HIV Agents--chemical synthesis Chelating Agents--pharmacology Chemistry, Pharmaceutical--methods Drug Design HIV Infections--drug therapy HIV Integrase Inhibitors--chemical synthesis Humans Metals--chemistry Models, Chemical Molecular Structure Naphthyridines--chemical synthesis Oxadiazoles--chemistry Structure-Activity Relationship Triazoles--chemistry