Li, Guo

14-O-Heterocyclic-substituted naltrexone derivatives as non-peptide mu opioid receptor selective antagonists: design, synthesis, and biological studies. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2009 - 1825-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2008.12.093 doi


Binding, Competitive
Chemistry, Pharmaceutical--methods
Drug Design
Humans
Kinetics
Ligands
Molecular Conformation
Molecular Structure
Naltrexone--analogs & derivatives
Narcotic Antagonists--chemical synthesis
Nitrogen--chemistry
Peptides--chemistry
Protein Structure, Tertiary
Receptors, Opioid, mu--antagonists & inhibitors