Calleja, Véronique

Role of a novel PH-kinase domain interface in PKB/Akt regulation: structural mechanism for allosteric inhibition. [electronic resource] - PLoS biology Jan 2009 - e17 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1545-7885

10.1371/journal.pbio.1000017 doi


3-Phosphoinositide-Dependent Protein Kinases
Allosteric Regulation--physiology
Animals
Binding Sites--drug effects
Gene Expression Regulation
Mice
Mutagenesis
Phosphorylation
Protein Conformation--drug effects
Protein Kinase Inhibitors--pharmacology
Protein Serine-Threonine Kinases--metabolism
Proto-Oncogene Proteins c-akt--antagonists & inhibitors
Structure-Activity Relationship