Sakurama, Kazufumi

Inhibition of focal adhesion kinase as a potential therapeutic strategy for imatinib-resistant gastrointestinal stromal tumor. [electronic resource] - Molecular cancer therapeutics Jan 2009 - 127-34 p. digital

Publication Type: Journal Article

1535-7163

10.1158/1535-7163.MCT-08-0884 doi


Administration, Oral
Animals
Benzamides
Cell Line
Cell Proliferation--drug effects
Drug Resistance, Neoplasm--drug effects
Female
Focal Adhesion Protein-Tyrosine Kinases--antagonists & inhibitors
Gastrointestinal Stromal Tumors--drug therapy
Imatinib Mesylate
Mice
Mice, Nude
Morpholines--administration & dosage
Mutation--genetics
Piperazines--therapeutic use
Proto-Oncogene Proteins c-akt--metabolism
Proto-Oncogene Proteins c-kit--genetics
Pyrimidines--therapeutic use
Substrate Specificity