Sidique, Shyama

Design and synthesis of pyrazole derivatives as potent and selective inhibitors of tissue-nonspecific alkaline phosphatase (TNAP). [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2009 - 222-5 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1464-3405

10.1016/j.bmcl.2008.10.107 doi


Alkaline Phosphatase--antagonists & inhibitors
Drug Design
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Humans
Inhibitory Concentration 50
Kinetics
Pyrazoles--chemical synthesis