Design and synthesis of pyrazole derivatives as potent and selective inhibitors of tissue-nonspecific alkaline phosphatase (TNAP). [electronic resource]
- Bioorganic & medicinal chemistry letters Jan 2009
- 222-5 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1464-3405
10.1016/j.bmcl.2008.10.107 doi
Alkaline Phosphatase--antagonists & inhibitors Drug Design Drug Evaluation, Preclinical Enzyme Inhibitors--chemical synthesis Humans Inhibitory Concentration 50 Kinetics Pyrazoles--chemical synthesis