Pichota, Arkadius
Peptide deformylase inhibitors of Mycobacterium tuberculosis: synthesis, structural investigations, and biological results. [electronic resource]
- Bioorganic & medicinal chemistry letters Dec 2008
- 6568-72 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2008.10.040 doi
Amidohydrolases--antagonists & inhibitors
Antitubercular Agents--chemistry
Chemistry, Pharmaceutical--methods
Crystallography, X-Ray--methods
Drug Design
Drug Resistance, Multiple
Fluoroquinolones--pharmacology
Gatifloxacin
Humans
Inhibitory Concentration 50
Microbial Sensitivity Tests
Models, Chemical
Molecular Conformation
Mycobacterium bovis--metabolism
Mycobacterium tuberculosis--drug effects
Tuberculosis--drug therapy