Pichota, Arkadius

Peptide deformylase inhibitors of Mycobacterium tuberculosis: synthesis, structural investigations, and biological results. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2008 - 6568-72 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2008.10.040 doi


Amidohydrolases--antagonists & inhibitors
Antitubercular Agents--chemistry
Chemistry, Pharmaceutical--methods
Crystallography, X-Ray--methods
Drug Design
Drug Resistance, Multiple
Fluoroquinolones--pharmacology
Gatifloxacin
Humans
Inhibitory Concentration 50
Microbial Sensitivity Tests
Models, Chemical
Molecular Conformation
Mycobacterium bovis--metabolism
Mycobacterium tuberculosis--drug effects
Tuberculosis--drug therapy