Design, synthesis, and evaluation of orally active inhibitors of plasminogen activator inhibitor-1 (PAI-1) production. [electronic resource]
- Bioorganic & medicinal chemistry letters Dec 2008
- 6419-22 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2008.10.067 doi
Administration, Oral Animals Benzylidene Compounds--chemical synthesis Biological Availability Chemistry, Pharmaceutical--methods Dogs Drug Administration Routes Drug Design Drug Evaluation, Preclinical Humans Models, Chemical Plasminogen Activator Inhibitor 1--chemistry Rats Solubility Succinimides--chemical synthesis