Muraglia, Ester

2-Trifluoroacetylthiophene oxadiazoles as potent and selective class II human histone deacetylase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2008 - 6083-7 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2008.09.076 doi


Combinatorial Chemistry Techniques
Drug Design
HCT116 Cells
Histone Acetyltransferases--antagonists & inhibitors
Histone Deacetylase Inhibitors
Histone Deacetylases--classification
Humans
Molecular Structure
Oxadiazoles--chemical synthesis
Structure-Activity Relationship
Thiophenes--chemical synthesis