Chao, Esther Y

Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity. [electronic resource] - Journal of medicinal chemistry Sep 2008 - 5758-65 p. digital

Publication Type: Journal Article

1520-4804

10.1021/jm800612u doi


Amines--chemistry
Anti-Inflammatory Agents--chemistry
Crystallography, X-Ray
DNA-Binding Proteins--drug effects
Drug Design
Liver X Receptors
Magnetic Resonance Spectroscopy
Mass Spectrometry
Models, Molecular
Molecular Structure
Orphan Nuclear Receptors
Receptors, Cytoplasmic and Nuclear--drug effects
Structure-Activity Relationship