Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity. [electronic resource]
- Journal of medicinal chemistry Sep 2008
- 5758-65 p. digital
Publication Type: Journal Article
1520-4804
10.1021/jm800612u doi
Amines--chemistry Anti-Inflammatory Agents--chemistry Crystallography, X-Ray DNA-Binding Proteins--drug effects Drug Design Liver X Receptors Magnetic Resonance Spectroscopy Mass Spectrometry Models, Molecular Molecular Structure Orphan Nuclear Receptors Receptors, Cytoplasmic and Nuclear--drug effects Structure-Activity Relationship