Nilsson, Johanna

Bupivacaine blocks N-type inactivating Kv channels in the open state: no allosteric effect on inactivation kinetics. [electronic resource] - Biophysical journal Dec 2008 - 5138-52 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1542-0086

10.1529/biophysj.108.130518 doi


Allosteric Regulation--drug effects
Animals
Binding Sites
Bupivacaine--pharmacology
Ion Channel Gating--drug effects
Kinetics
Models, Molecular
Potassium Channel Blockers--pharmacology
Potassium Channels, Voltage-Gated--metabolism
Shaw Potassium Channels--metabolism
Time Factors
Xenopus Proteins--metabolism
Xenopus laevis--metabolism