TY - GEN AU - Tong,Yunsong AU - Stewart,Kent D AU - Thomas,Sheela AU - Przytulinska,Magdalena AU - Johnson,Eric F AU - Klinghofer,Vered AU - Leverson,Joel AU - McCall,Owen AU - Soni,Niru B AU - Luo,Yan AU - Lin,Nan-horng AU - Sowin,Thomas J AU - Giranda,Vincent L AU - Penning,Thomas D TI - Isoxazolo[3,4-b]quinoline-3,4(1H,9H)-diones as unique, potent and selective inhibitors for Pim-1 and Pim-2 kinases: chemistry, biological activities, and molecular modeling SN - 1464-3405 PY - 2008///1030 KW - Combinatorial Chemistry Techniques KW - Crystallography, X-Ray KW - Humans KW - Isoxazoles KW - chemical synthesis KW - Models, Molecular KW - Molecular Conformation KW - Molecular Structure KW - Protein Serine-Threonine Kinases KW - antagonists & inhibitors KW - Proto-Oncogene Proteins KW - Proto-Oncogene Proteins c-pim-1 KW - Quinolines KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2008.08.079 ER -