Synthesis of anti-microtubule biaryls and preliminary evaluation as vascular-disrupting agents. [electronic resource]
- ChemMedChem Nov 2008
- 1731-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1860-7187
10.1002/cmdc.200800181 doi
Angiogenesis Inhibitors--pharmacology Cell Line, Tumor Cell Proliferation Cells, Cultured Chemistry, Pharmaceutical--methods Drug Design Endothelial Cells--metabolism Endothelium, Vascular--drug effects Humans Inhibitory Concentration 50 Ligands Magnetic Resonance Spectroscopy Microtubules--chemistry Models, Chemical Tubulin--chemistry