Tarragó, Teresa Baicalin, a prodrug able to reach the CNS, is a prolyl oligopeptidase inhibitor. [electronic resource] - Bioorganic & medicinal chemistry Aug 2008 - 7516-24 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1464-3391 Standard No.: 10.1016/j.bmc.2008.04.067 doi Subjects--Topical Terms: Dose-Response Relationship, DrugEnzyme Inhibitors--chemistryFlavanones--chemistryFlavonoids--chemistryProlyl OligopeptidasesSerine Endopeptidases--metabolismStructure-Activity Relationship