Zientek, Michael

Development of an in vitro drug-drug interaction assay to simultaneously monitor five cytochrome P450 isoforms and performance assessment using drug library compounds. [electronic resource] - Journal of pharmacological and toxicological methods - 206-14 p. digital

Publication Type: Journal Article

1873-488X

10.1016/j.vascn.2008.05.131 doi


Aryl Hydrocarbon Hydroxylases--metabolism
Chromatography, Liquid--methods
Cytochrome P-450 CYP1A2--metabolism
Cytochrome P-450 CYP2C9
Cytochrome P-450 Enzyme System--metabolism
Dextromethorphan--metabolism
Diclofenac--metabolism
Drug Interactions
Humans
Isoenzymes--metabolism
Mass Spectrometry--methods
Mephenytoin--metabolism
Miconazole--metabolism
Microsomes, Liver--drug effects
Midazolam--metabolism
Substrate Specificity
Tacrine--metabolism
Testosterone--metabolism