Cyclooxygenase inhibitors down regulate P-glycoprotein in human colorectal Caco-2 cell line. [electronic resource]
- Pharmaceutical research Sep 2008
- 1991-2001 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0724-8741
10.1007/s11095-008-9596-1 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--genetics Antineoplastic Agents--pharmacology Caco-2 Cells Celecoxib Colorectal Neoplasms--drug therapy Cyclooxygenase 1--metabolism Cyclooxygenase 2--metabolism Cyclooxygenase 2 Inhibitors--pharmacology Dinoprostone--metabolism Down-Regulation Drug Resistance, Neoplasm--drug effects Gene Expression Regulation, Neoplastic--drug effects Humans Indomethacin--analogs & derivatives Naproxen--pharmacology Neoplasm Proteins--genetics Pyrazoles--pharmacology RNA, Messenger--metabolism Reproducibility of Results Sulfonamides--pharmacology Time Factors