Shah, Unmesh

Biaryl and heteroaryl derivatives of SCH 58261 as potent and selective adenosine A2A receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Jul 2008 - 4199-203 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2008.05.074 doi


Adenosine A2 Receptor Antagonists
Administration, Oral
Animals
Behavior, Animal--drug effects
Chemistry, Pharmaceutical--methods
Drug Design
Humans
Models, Chemical
Neuroprotective Agents--chemical synthesis
Parkinson Disease--drug therapy
Piperazines--chemistry
Pyrimidines--chemical synthesis
Quinolines--chemistry
Rats
Structure-Activity Relationship
Triazoles--chemical synthesis