TY - GEN AU - Kreft,Anthony AU - Harrison,Boyd AU - Aschmies,Suzan AU - Atchison,Kevin AU - Casebier,David AU - Cole,Derek C AU - Diamantidis,George AU - Ellingboe,John AU - Hauze,Diane AU - Hu,Yun AU - Huryn,Donna AU - Jin,Mei AU - Kubrak,Dennis AU - Lu,Peimin AU - Lundquist,Joseph AU - Mann,Charles AU - Martone,Robert AU - Moore,William AU - Oganesian,Aram AU - Porte,Alex AU - Riddell,Dave R AU - Sonnenberg-Reines,June AU - Stock,Joseph R AU - Sun,Shaiu-Ching AU - Wagner,Erik AU - Woller,Kevin AU - Xu,Zheng AU - Zhou,Hua AU - Steven Jacobsen,J TI - Discovery of a novel series of Notch-sparing gamma-secretase inhibitors SN - 1464-3405 PY - 2008///1117 KW - Alzheimer Disease KW - drug therapy KW - Amyloid KW - chemistry KW - Amyloid Precursor Protein Secretases KW - antagonists & inhibitors KW - Carbon KW - Chemistry, Pharmaceutical KW - methods KW - Drug Design KW - Drug Evaluation, Preclinical KW - Enzyme Inhibitors KW - chemical synthesis KW - Humans KW - Models, Chemical KW - Receptors, Notch KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2008.05.064 ER -