Discovery of a novel series of Notch-sparing gamma-secretase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Jul 2008
- 4232-6 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2008.05.064 doi
Alzheimer Disease--drug therapy Amyloid--chemistry Amyloid Precursor Protein Secretases--antagonists & inhibitors Carbon--chemistry Chemistry, Pharmaceutical--methods Drug Design Drug Evaluation, Preclinical Enzyme Inhibitors--chemical synthesis Humans Models, Chemical Receptors, Notch--antagonists & inhibitors Structure-Activity Relationship