Discovery of a novel class of 2-ureido thiophene carboxamide checkpoint kinase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Jul 2008
- 4242-8 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2008.05.016 doi
Amides--chemistry Apoptosis Carbon--chemistry Cell Cycle Checkpoint Kinase 1 Chemistry, Pharmaceutical--methods DNA Damage Drug Design Humans Inhibitory Concentration 50 Models, Chemical Phenyl Ethers--chemistry Protein Kinase Inhibitors--chemical synthesis Protein Kinases--chemistry Thiophenes--chemistry Urea--chemistry