Discovery and characterization of QPT-1, the progenitor of a new class of bacterial topoisomerase inhibitors. [electronic resource]
- Antimicrobial agents and chemotherapy Aug 2008
- 2806-12 p. digital
Publication Type: Journal Article
1098-6596
10.1128/AAC.00247-08 doi
Animals Anti-Bacterial Agents--chemistry Area Under Curve Bacteria--drug effects Bacterial Infections--metabolism Bacterial Proteins--antagonists & inhibitors Cell Line Cell Proliferation--drug effects Metabolic Clearance Rate Mice Microbial Sensitivity Tests Molecular Structure Staphylococcus aureus--drug effects Stereoisomerism Topoisomerase II Inhibitors