TY - GEN AU - Guo,Jianxia AU - Parise,Robert A AU - Joseph,Erin AU - Egorin,Merrill J AU - Lazo,John S AU - Prochownik,Edward V AU - Eiseman,Julie L TI - Efficacy, pharmacokinetics, tisssue distribution, and metabolism of the Myc-Max disruptor, 10058-F4 [Z,E]-5-[4-ethylbenzylidine]-2-thioxothiazolidin-4-one, in mice SN - 1432-0843 PY - 2009///0331 KW - Animals KW - Basic Helix-Loop-Helix Leucine Zipper Transcription Factors KW - antagonists & inhibitors KW - Cell Proliferation KW - drug effects KW - Chromatography, High Pressure Liquid KW - Chromatography, Liquid KW - Dimerization KW - Female KW - Humans KW - Male KW - Mice KW - Mice, SCID KW - Prostatic Neoplasms KW - drug therapy KW - Proto-Oncogene Proteins c-myc KW - Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization KW - Thiazoles KW - pharmacokinetics KW - Tissue Distribution KW - Treatment Outcome KW - Tumor Cells, Cultured KW - Xenograft Model Antitumor Assays N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S UR - https://doi.org/10.1007/s00280-008-0774-y ER -