Wolin, Ronald L
Dual binding site inhibitors of B-RAF kinase. [electronic resource]
- Bioorganic & medicinal chemistry letters May 2008
- 2825-9 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2008.04.002 doi
Adenosine Triphosphate--metabolism
Allosteric Site
Computer-Aided Design
Crystallography, X-Ray
Extracellular Signal-Regulated MAP Kinases--antagonists & inhibitors
Hydrocarbons, Aromatic--chemical synthesis
Imidazoles--chemical synthesis
Inhibitory Concentration 50
Phosphorylation--drug effects
Protein Kinase Inhibitors--chemical synthesis
Proto-Oncogene Proteins B-raf--antagonists & inhibitors
Structure-Activity Relationship