TY - GEN AU - Ward,Simon E AU - Eddershaw,Peter J AU - Scott,Claire M AU - Gordon,Laurie J AU - Lovell,Peter J AU - Moore,Susan H AU - Smith,Paul W AU - Starr,Kathryn R AU - Thewlis,Kevin M AU - Watson,Jeannette M TI - Discovery of potent, orally bioavailable, selective 5-HT1A/B/D receptor antagonists SN - 0022-2623 PY - 2008///0709 KW - Animals KW - Blood-Brain Barrier KW - metabolism KW - Cerebral Cortex KW - Humans KW - In Vitro Techniques KW - Piperazines KW - chemical synthesis KW - Quinolines KW - Radioligand Assay KW - Rats KW - Recombinant Proteins KW - pharmacology KW - Serotonin 5-HT1 Receptor Antagonists KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/jm8001444 ER -