Ward, Simon E Discovery of potent, orally bioavailable, selective 5-HT1A/B/D receptor antagonists. [electronic resource] - Journal of medicinal chemistry May 2008 - 2887-90 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm8001444 doi Subjects--Topical Terms: AnimalsBlood-Brain Barrier--metabolismCerebral Cortex--metabolismHumansIn Vitro TechniquesPiperazines--chemical synthesisQuinolines--chemical synthesisRadioligand AssayRatsRecombinant Proteins--pharmacologySerotonin 5-HT1 Receptor AntagonistsStructure-Activity Relationship