LPK-26, a novel kappa-opioid receptor agonist with potent antinociceptive effects and low dependence potential. [electronic resource]
- European journal of pharmacology Apr 2008
- 306-11 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0014-2999
10.1016/j.ejphar.2008.02.028 doi
Acetic Acid Analgesics, Opioid--pharmacology Animals Behavior, Animal--drug effects CHO Cells Cricetinae Cricetulus Disease Models, Animal Dose-Response Relationship, Drug Guanosine 5'-O-(3-Thiotriphosphate)--metabolism Hot Temperature--adverse effects Humans Male Mice Motor Activity--drug effects Naloxone--pharmacology Narcotic Antagonists--pharmacology Opioid-Related Disorders--prevention & control Pain--etiology Pain Measurement Pain Threshold--drug effects Protein Binding Pyrroles--pharmacology Rats Receptors, Opioid, delta--agonists Receptors, Opioid, kappa--agonists Receptors, Opioid, mu--agonists Time Factors Transfection