Design and synthesis of dual inhibitors of HIV reverse transcriptase and integrase: introducing a diketoacid functionality into delavirdine. [electronic resource]
- Bioorganic & medicinal chemistry Apr 2008
- 3587-95 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2008.02.007 doi
Delavirdine--chemistry Drug Design HIV--drug effects HIV Integrase--metabolism HIV Integrase Inhibitors--chemical synthesis HIV Reverse Transcriptase--antagonists & inhibitors Keto Acids--chemistry Molecular Structure Reverse Transcriptase Inhibitors--chemical synthesis