Kim, Y W

Pharmacokinetics and tissue distribution of 3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methyl)benzamide; a novel ALK5 inhibitor and a potential anti-fibrosis drug. [electronic resource] - Xenobiotica; the fate of foreign compounds in biological systems Mar 2008 - 325-39 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0049-8254

10.1080/00498250701781924 doi


Administration, Oral
Animals
Benzamides--administration & dosage
Biological Transport--drug effects
Caco-2 Cells
Chromatography, Liquid
Dogs
Enzyme Inhibitors--administration & dosage
Half-Life
Haplorhini
Humans
Imidazoles--administration & dosage
Injections, Intravenous
Magnetic Resonance Spectroscopy
Male
Mass Spectrometry
Mice
Models, Biological
Protein Serine-Threonine Kinases--antagonists & inhibitors
Quinoxalines--administration & dosage
Rats
Rats, Sprague-Dawley
Receptor, Transforming Growth Factor-beta Type I
Receptors, Transforming Growth Factor beta--antagonists & inhibitors
Tissue Distribution--drug effects