Potent, exceptionally selective, orally bioavailable inhibitors of TNF-alpha Converting Enzyme (TACE): novel 2-substituted-1H-benzo[d]imidazol-1-yl)methyl)benzamide P1' substituents. [electronic resource]
- Bioorganic & medicinal chemistry letters Mar 2008
- 1577-82 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2008.01.075 doi
ADAM Proteins--antagonists & inhibitors ADAM17 Protein Animals Area Under Curve Benzamides--blood Biological Availability Dogs Half-Life Molecular Structure Rats Structure-Activity Relationship