Fu, Kai

SM16, an orally active TGF-beta type I receptor inhibitor prevents myofibroblast induction and vascular fibrosis in the rat carotid injury model. [electronic resource] - Arteriosclerosis, thrombosis, and vascular biology Apr 2008 - 665-71 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1524-4636

10.1161/ATVBAHA.107.158030 doi


Activin Receptors, Type I--antagonists & inhibitors
Adenosine Triphosphate--metabolism
Administration, Oral
Animals
Azabicyclo Compounds--administration & dosage
Binding Sites
Carotid Artery Injuries--drug therapy
Cell Line
Fibroblasts--drug effects
Fibrosis
Humans
Male
Myoblasts, Smooth Muscle--drug effects
Protein Kinase Inhibitors--administration & dosage
Protein Serine-Threonine Kinases--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Receptor, Transforming Growth Factor-beta Type I
Receptors, Transforming Growth Factor beta--antagonists & inhibitors
Transforming Growth Factor beta--physiology