Development and implementation of a miniaturized high-throughput time-resolved fluorescence energy transfer assay to identify small molecule inhibitors of polo-like kinase 1. [electronic resource]
- Assay and drug development technologies Dec 2007
- 723-35 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1540-658X
10.1089/adt.2007.102 doi
Blotting, Western Cell Cycle Proteins--antagonists & inhibitors Data Interpretation, Statistical Drug Design Drug Evaluation, Preclinical Enzyme Inhibitors--chemical synthesis Fluorescence Resonance Energy Transfer Fluorometry Freezing Hydrogen-Ion Concentration Indicators and Reagents Kinetics Miniaturization Protein Kinase C--antagonists & inhibitors Protein Serine-Threonine Kinases--antagonists & inhibitors Proto-Oncogene Proteins--antagonists & inhibitors Reproducibility of Results Silver Staining Substrate Specificity Temperature Polo-Like Kinase 1