Sharlow, Elizabeth R

Development and implementation of a miniaturized high-throughput time-resolved fluorescence energy transfer assay to identify small molecule inhibitors of polo-like kinase 1. [electronic resource] - Assay and drug development technologies Dec 2007 - 723-35 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1540-658X

10.1089/adt.2007.102 doi


Blotting, Western
Cell Cycle Proteins--antagonists & inhibitors
Data Interpretation, Statistical
Drug Design
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Fluorescence Resonance Energy Transfer
Fluorometry
Freezing
Hydrogen-Ion Concentration
Indicators and Reagents
Kinetics
Miniaturization
Protein Kinase C--antagonists & inhibitors
Protein Serine-Threonine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins--antagonists & inhibitors
Reproducibility of Results
Silver Staining
Substrate Specificity
Temperature
Polo-Like Kinase 1