De La Fuente, Ricardo Small-molecule screen identifies inhibitors of a human intestinal calcium-activated chloride channel. [electronic resource] - Molecular pharmacology Mar 2008 - 758-68 p. digital Publication Type: Journal Article; Research Support, N.I.H., Extramural ISSN: 1521-0111 Standard No.: 10.1124/mol.107.043208 doi Subjects--Topical Terms: Adenosine Triphosphate--antagonists & inhibitorsCalcium--analysisCarbachol--antagonists & inhibitorsChloride Channels--antagonists & inhibitorsChlorides--metabolismDose-Response Relationship, DrugDrug Evaluation, Preclinical--methodsFluorescent Dyes--metabolismFura-2--metabolismGenetic VectorsHT29 CellsHumansInhibitory Concentration 50Intestinal Mucosa--metabolismIntestines--drug effectsIon Channel Gating--drug effectsKineticsLentivirus--geneticsModels, BiologicalMolecular StructurePatch-Clamp TechniquesReproducibility of ResultsStructure-Activity Relationship