De La Fuente, Ricardo

Small-molecule screen identifies inhibitors of a human intestinal calcium-activated chloride channel. [electronic resource] - Molecular pharmacology Mar 2008 - 758-68 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1521-0111

10.1124/mol.107.043208 doi


Adenosine Triphosphate--antagonists & inhibitors
Calcium--analysis
Carbachol--antagonists & inhibitors
Chloride Channels--antagonists & inhibitors
Chlorides--metabolism
Dose-Response Relationship, Drug
Drug Evaluation, Preclinical--methods
Fluorescent Dyes--metabolism
Fura-2--metabolism
Genetic Vectors
HT29 Cells
Humans
Inhibitory Concentration 50
Intestinal Mucosa--metabolism
Intestines--drug effects
Ion Channel Gating--drug effects
Kinetics
Lentivirus--genetics
Models, Biological
Molecular Structure
Patch-Clamp Techniques
Reproducibility of Results
Structure-Activity Relationship