Iwamoto, Marian
Lack of a pharmacokinetic effect of raltegravir on midazolam: in vitro/in vivo correlation. [electronic resource]
- Journal of clinical pharmacology Feb 2008
- 209-14 p. digital
Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
ISSN: 0091-2700
Standard No.: 10.1177/0091270007310382 doi
Subjects--Topical Terms: Area Under Curve Cells, Cultured Chromatography, Liquid Cross-Over Studies Cytochrome P-450 CYP3A--genetics Dose-Response Relationship, Drug Drug Interactions Female HIV Integrase Inhibitors--pharmacology Half-Life Hepatocytes--cytology Humans Male Mass Spectrometry Metabolic Clearance Rate Microsomes, Liver--drug effects Midazolam--administration & dosage Organic Chemicals--pharmacology Pyrrolidinones Raltegravir Potassium Reverse Transcriptase Polymerase Chain Reaction