TY - GEN AU - Douty,Brent AU - Wayland,Brian AU - Ala,Paul J AU - Bower,Michael J AU - Pruitt,James AU - Bostrom,Lori AU - Wei,Min AU - Klabe,Ronald AU - Gonneville,Lucie AU - Wynn,Richard AU - Burn,Timothy C AU - Liu,Phillip C C AU - Combs,Andrew P AU - Yue,Eddy W TI - Isothiazolidinone inhibitors of PTP1B containing imidazoles and imidazolines SN - 1464-3405 PY - 2008///0212 KW - Crystallography, X-Ray KW - Drug Design KW - Enzyme Inhibitors KW - chemical synthesis KW - Imidazoles KW - Imidazolines KW - Models, Molecular KW - Protein Tyrosine Phosphatase, Non-Receptor Type 1 KW - antagonists & inhibitors KW - Structure-Activity Relationship KW - Thiazoles N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2007.11.012 ER -