Design and characterization of bivalent Smac-based peptides as antagonists of XIAP and development and validation of a fluorescence polarization assay for XIAP containing both BIR2 and BIR3 domains. [electronic resource]
- Analytical biochemistry Mar 2008
- 87-98 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.; Validation Study
0003-2697
10.1016/j.ab.2007.10.032 doi
Apoptosis Regulatory Proteins Biomimetic Materials--chemical synthesis Caspase Inhibitors Chromatography, Gel Fluorescence Polarization--methods Humans Intracellular Signaling Peptides and Proteins--chemical synthesis Kinetics Ligands Mitochondrial Proteins--chemical synthesis Oligopeptides--chemical synthesis Protein Binding Protein Structure, Tertiary X-Linked Inhibitor of Apoptosis Protein--analysis