TY - GEN AU - Sabbatini,Fabio Maria AU - Di Fabio,Romano AU - St-Denis,Yves AU - Capelli,Anna-Maria AU - Castiglioni,Emiliano AU - Contini,Stefania AU - Donati,Daniele AU - Fazzolari,Elettra AU - Gentile,Gabriella AU - Micheli,Fabrizio AU - Pavone,Francesca AU - Rinaldi,Marilisa AU - Pasquarello,Alessandra AU - Zampori,Maria Grazia AU - Di Felice,Pina AU - Zarantonello,Paola AU - Arban,Roberto AU - Perini,Benedetta AU - Vitulli,Giovanni AU - Benedetti,Roberto AU - Oliosi,Beatrice AU - Worby,Angela TI - Heteroaryl-substituted 4-(1H-pyrazol-1-yl)-5,6-dihydro-1H-pyrrolo[2,3-d]pyrimidine derivatives as potent and selective corticotropin-releasing factor receptor-1 antagonists SN - 1860-7187 PY - 2008///0723 KW - Animals KW - Anxiety KW - drug therapy KW - Corticotropin-Releasing Hormone KW - metabolism KW - Depression KW - Drug Design KW - Models, Chemical KW - Pyrazoles KW - chemical synthesis KW - Pyrimidines KW - Rats KW - Rats, Wistar KW - Receptors, Corticotropin-Releasing Hormone KW - antagonists & inhibitors KW - Structure-Activity Relationship KW - CRF Receptor, Type 1 N1 - Publication Type: Journal Article UR - https://doi.org/10.1002/cmdc.200700230 ER -