Sabbatini, Fabio Maria

Heteroaryl-substituted 4-(1H-pyrazol-1-yl)-5,6-dihydro-1H-pyrrolo[2,3-d]pyrimidine derivatives as potent and selective corticotropin-releasing factor receptor-1 antagonists. [electronic resource] - ChemMedChem Feb 2008 - 226-9 p. digital

Publication Type: Journal Article

1860-7187

10.1002/cmdc.200700230 doi


Animals
Anxiety--drug therapy
Corticotropin-Releasing Hormone--metabolism
Depression--drug therapy
Drug Design
Models, Chemical
Pyrazoles--chemical synthesis
Pyrimidines--chemical synthesis
Rats
Rats, Wistar
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Structure-Activity Relationship
CRF Receptor, Type 1