Angell, Richard M

Biphenyl amide p38 kinase inhibitors 2: Optimisation and SAR. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2008 - 324-8 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2007.10.043 doi


Administration, Oral
Amides--chemistry
Animals
Arthritis, Experimental--drug therapy
Biphenyl Compounds--chemistry
Crystallography, X-Ray
Models, Molecular
Molecular Conformation
Oxadiazoles--chemistry
Piperazines--chemistry
Protein Binding
Protein Kinase Inhibitors--chemistry
Rats
Structure-Activity Relationship
p38 Mitogen-Activated Protein Kinases--antagonists & inhibitors