Angell, Richard M
Biphenyl amide p38 kinase inhibitors 2: Optimisation and SAR. [electronic resource]
- Bioorganic & medicinal chemistry letters Jan 2008
- 324-8 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2007.10.043 doi
Administration, Oral
Amides--chemistry
Animals
Arthritis, Experimental--drug therapy
Biphenyl Compounds--chemistry
Crystallography, X-Ray
Models, Molecular
Molecular Conformation
Oxadiazoles--chemistry
Piperazines--chemistry
Protein Binding
Protein Kinase Inhibitors--chemistry
Rats
Structure-Activity Relationship
p38 Mitogen-Activated Protein Kinases--antagonists & inhibitors