TY  - GEN
AU  - Cole,Derek C
AU  - Stock,Joseph R
AU  - Lennox,William J
AU  - Bernotas,Ronald C
AU  - Ellingboe,John W
AU  - Boikess,Steve
AU  - Coupet,Joseph
AU  - Smith,Deborah L
AU  - Leung,Louis
AU  - Zhang,Guo-Ming
AU  - Feng,Xidong
AU  - Kelly,Michael F
AU  - Galante,Rocco
AU  - Huang,Pingzhong
AU  - Dawson,Lee A
AU  - Marquis,Karen
AU  - Rosenzweig-Lipson,Sharon
AU  - Beyer,Chad E
AU  - Schechter,Lee E
TI  - Discovery of N1-(6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonyl)tryptamine as a potent, selective, and orally active 5-HT(6) receptor agonist
SN  - 0022-2623
PY  - 2008///0108
KW  - Administration, Oral
KW  - Animals
KW  - Biological Availability
KW  - CHO Cells
KW  - Cricetinae
KW  - Cricetulus
KW  - Dogs
KW  - Frontal Lobe
KW  - metabolism
KW  - Haplorhini
KW  - Humans
KW  - In Vitro Techniques
KW  - Mice
KW  - Microdialysis
KW  - Microsomes, Liver
KW  - Radioligand Assay
KW  - Rats
KW  - Receptors, Serotonin
KW  - Serotonin Receptor Agonists
KW  - chemical synthesis
KW  - Solubility
KW  - Structure-Activity Relationship
KW  - Thiazoles
KW  - chemistry
KW  - Tryptamines
KW  - gamma-Aminobutyric Acid
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1021/jm070521y
ER  -