Venneti, Sriram

The high affinity peripheral benzodiazepine receptor ligand DAA1106 binds to activated and infected brain macrophages in areas of synaptic degeneration: implications for PET imaging of neuroinflammation in lentiviral encephalitis. [electronic resource] - Neurobiology of disease Feb 2008 - 232-41 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

0969-9961

10.1016/j.nbd.2007.08.016 doi


Acetamides--pharmacokinetics
Adult
Aged
Analysis of Variance
Animals
Antigens, CD--metabolism
Antigens, Differentiation, Myelomonocytic--metabolism
Astrocytes--drug effects
Brain--diagnostic imaging
Bucladesine--pharmacology
Dose-Response Relationship, Drug
Encephalitis, Viral--pathology
Female
Humans
Lentivirus
Lipopolysaccharides--pharmacology
Macaca mulatta
Macrophages--drug effects
Male
Middle Aged
Nerve Tissue Proteins--metabolism
Phenyl Ethers--pharmacokinetics
Positron-Emission Tomography
Protein Binding--drug effects
Synapses--drug effects