Knör, Sebastian

Development and evaluation of peptidic ligands targeting tumour-associated urokinase plasminogen activator receptor (uPAR) for use in alpha-emitter therapy for disseminated ovarian cancer. [electronic resource] - European journal of nuclear medicine and molecular imaging Jan 2008 - 53-64 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1619-7089

10.1007/s00259-007-0582-3 doi


Alpha Particles--therapeutic use
Animals
Bismuth--chemistry
Cell Line, Tumor
Dimerization
Drug Discovery
Enzyme Inhibitors--chemistry
Female
Gene Expression Regulation, Neoplastic
Heterocyclic Compounds, 1-Ring--chemistry
Humans
Kidney--drug effects
Ligands
Mice
Neoplasm Metastasis
Ovarian Neoplasms--genetics
Peptides--chemical synthesis
Polygeline--pharmacology
Radioisotopes
Receptors, Urokinase Plasminogen Activator--antagonists & inhibitors
Solubility
Substrate Specificity
Tissue Distribution