Micheli, Fabrizio
1,2,4-triazol-3-yl-thiopropyl-tetrahydrobenzazepines: a series of potent and selective dopamine D(3) receptor antagonists. [electronic resource]
- Journal of medicinal chemistry Oct 2007
- 5076-89 p. digital
Publication Type: Journal Article
ISSN: 0022-2623
Standard No.: 10.1021/jm0705612 doi
Subjects--Topical Terms: Acetylcholine--metabolism Administration, Oral Alcohol Drinking--prevention & control Animals Benzazepines--chemical synthesis Brain--blood supply Cocaine--pharmacology Conditioning, Operant--drug effects ERG1 Potassium Channel Ether-A-Go-Go Potassium Channels--metabolism Guinea Pigs Histamine H1 Antagonists--chemical synthesis Humans In Vitro Techniques Male Mice Mice, Inbred C57BL Microsomes, Liver--drug effects Models, Molecular Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Dopamine D3--agonists Receptors, Histamine H1--metabolism Structure-Activity Relationship Tobacco Use Disorder--prevention & control Triazoles--chemical synthesis