Discovery of 4'-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-benzonitriles and 4'-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-pyridine-2'-carbonitriles as potent checkpoint kinase 1 (Chk1) inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Nov 2007
- 5944-51 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2007.07.102 doi
Checkpoint Kinase 1 Nitriles--chemistry Protein Kinase Inhibitors--chemistry Protein Kinases--drug effects Structure-Activity Relationship