Tao, Zhi-Fu

Discovery of 4'-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-benzonitriles and 4'-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-pyridine-2'-carbonitriles as potent checkpoint kinase 1 (Chk1) inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2007 - 5944-51 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2007.07.102 doi


Checkpoint Kinase 1
Nitriles--chemistry
Protein Kinase Inhibitors--chemistry
Protein Kinases--drug effects
Structure-Activity Relationship